GPCR CLASS (FAMILY)
Class A (Rhodopsin)
GPCR SPECIES
Homo sapiens
GPCR PREFERRED CHAIN
R
G PROTEIN (FAMILY)
Gq/11
G PROTEIN SPECIES
Homo sapiens
PDB CODE
RESOLUTION
3.1 Å
REFERENCE
PUBLICATION DATE
Aug. 9, 2023
LIGAND INTERACTIONS
LIGANDS
JMV431 - Agonist gtoplig chembl_ligand pubchem ,
CHEMBL4576388 - PAM chembl_ligand pubchem
PHYSIOLOGICAL LIGANDS
neurotensin, neuromedin N, large neurotensin, large neuromedin N