Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
aa2ar_human 146 ECL2 C => S Abolished EC50 (cAMP accumulation) adenosine De Filippo E et al (2016)
aa2ar_human 146 ECL2 C => S 7.343↑ EC50 (cAMP accumulation) NECA De Filippo E et al (2016)
aa2ar_human 146 ECL2 C => S 5.525↓ K(i) (radioligand binding) NECA De Filippo E et al (2016)
aa2ar_human 146 ECL2 C => S 25.421↑ EC50 (cAMP accumulation) CGS21680 De Filippo E et al (2016)
aa2ar_human 146 ECL2 C => S 1.095↓ K(i) (radioligand binding) CGS21680 De Filippo E et al (2016)
aa2ar_human 146 ECL2 C => S Abolished EC50 (cAMP accumulation) PSB-15826 De Filippo E et al (2016)
aa2ar_human 146 ECL2 C => S 1.283↑ K(i) (radioligand binding) PSB-15826 De Filippo E et al (2016)
aa2ar_human 159 ECL2 C => S 21.739↓ EC50 (cAMP accumulation) adenosine De Filippo E et al (2016)
aa2ar_human 159 ECL2 C => S 8.268↑ EC50 (cAMP accumulation) NECA De Filippo E et al (2016)
aa2ar_human 159 ECL2 C => S 4.02↑ K(i) (radioligand binding) NECA De Filippo E et al (2016)
aa2ar_human 159 ECL2 C => S 5.443↑ EC50 (cAMP accumulation) CGS21680 De Filippo E et al (2016)
aa2ar_human 159 ECL2 C => S 2.595↑ K(i) (radioligand binding) CGS21680 De Filippo E et al (2016)
aa2ar_human 159 ECL2 C => S 25.726↑ EC50 (cAMP accumulation) PSB-15826 De Filippo E et al (2016)
aa2ar_human 159 ECL2 C => S 4.041↑ K(i) (radioligand binding) PSB-15826 De Filippo E et al (2016)
aa2ar_human 45.50x50 166 ECL2 C => S 30.303↓ EC50 (cAMP accumulation) adenosine De Filippo E et al (2016)
aa2ar_human 45.50x50 166 ECL2 C => S 2.994↓ EC50 (cAMP accumulation) NECA De Filippo E et al (2016)
aa2ar_human 45.50x50 166 ECL2 C => S 1.224↓ K(i) (radioligand binding) NECA De Filippo E et al (2016)
aa2ar_human 45.50x50 166 ECL2 C => S 1.56↓ EC50 (cAMP accumulation) CGS21680 De Filippo E et al (2016)
aa2ar_human 45.50x50 166 ECL2 C => S 1.14↑ K(i) (radioligand binding) CGS21680 De Filippo E et al (2016)
aa2ar_human 45.50x50 166 ECL2 C => S 1.209↓ EC50 (cAMP accumulation) PSB-15826 De Filippo E et al (2016)
aa2ar_human 45.50x50 166 ECL2 C => S 1.661↓ K(i) (radioligand binding) PSB-15826 De Filippo E et al (2016)
aa2ar_human 6.55x55 253 TM6 N => Q N/A N/A Kim J et al (1995)
aa2ar_human 6.55x55 253 TM6 N => S N/A N/A Kim J et al (1995)
aa2ar_human 7.43x42 278 TM7 H => Q N/A N/A Kim J et al (1995)
aa2ar_human 7.43x42 278 TM7 H => F N/A N/A Kim J et al (1995)
aa2ar_human 7.43x42 278 TM7 H => Y N/A N/A Kim J et al (1995)
aa2ar_human 151 ECL2 E => A N/A N/A Kim J et al (1996)
aa2ar_human 151 ECL2 E => Q N/A N/A Kim J et al (1996)
aa2ar_human 151 ECL2 E => D N/A N/A Kim J et al (1996)
aa2ar_human 161 ECL2 E => A N/A N/A Kim J et al (1996)
aa2ar_human 169 ECL2 E => A N/A N/A Kim J et al (1996)
aa2ar_human 169 ECL2 E => Q N/A N/A Kim J et al (1996)
aa2ar_human 170 ECL2 D => K N/A N/A Kim J et al (1996)
aa2ar_human 5.34x36 173 TM5 P => R N/A N/A Kim J et al (1996)
aa2ar_human 262 ECL3 C => G N/A N/A Kim J et al (1996)
aa2ar_human 1.39x39 13 TM1 E => Q N/A N/A IJzerman AP et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.38x38 90 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 7.42x41 277 TM7 S => C N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => N N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => L N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => H N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => R N/A N/A Jiang Q et al (1996)
aa2ar_human 1.39x39 13 TM1 E => Q N/A N/A IJzerman AP et al (1996)
aa2ar_human 3.32x32 84 TM3 V => A N/A N/A Jiang Q et al (1997)
aa2ar_human 3.32x32 84 TM3 V => D N/A N/A Jiang Q et al (1997)
aa2ar_human 3.32x32 84 TM3 V => L N/A N/A Jiang Q et al (1997)
aa2ar_human 6.52x52 250 TM6 H => N N/A N/A Jiang Q et al (1997)
aa2ar_human 7.43x42 278 TM7 H => K N/A N/A Jiang Q et al (1997)
aa2ar_human 7.43x42 278 TM7 H => N N/A N/A Jiang Q et al (1997)
aa2ar_human 5.41x42 180 TM5 F => A N/A N/A Kim J et al (1995)
aa2ar_human 5.42x43 181 TM5 N => S N/A N/A Kim J et al (1995)
aa2ar_human 5.43x44 182 TM5 F => W N/A N/A Kim J et al (1995)
aa2ar_human 5.43x44 182 TM5 F => A N/A N/A Kim J et al (1995)
aa2ar_human 6.52x52 250 TM6 H => F N/A N/A Kim J et al (1995)
aa2ar_human 5.43x44 182 TM5 F => Y N/A N/A Kim J et al (1995)
aa2ar_human 6.52x52 250 TM6 H => A N/A N/A Kim J et al (1995)
aa2ar_human 6.52x52 250 TM6 H => Y N/A N/A Kim J et al (1995)
aa2ar_human 6.55x55 253 TM6 N => A N/A N/A Kim J et al (1995)
aa2ar_human 6.56x56 254 TM6 C => A N/A N/A Kim J et al (1995)
aa2ar_human 6.59x59 257 TM6 F => A N/A N/A Kim J et al (1995)
aa2ar_human 7.36x35 271 TM7 Y => A N/A N/A Kim J et al (1995)
aa2ar_human 7.39x38 274 TM7 I => A N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => A N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.43x42 278 TM7 H => A N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => A N/A N/A Kim J et al (1995)
aa2ar_human 1.39x39 13 TM1 E => Q N/A N/A Gao ZG et al (2000)
aa2ar_human 7.43x42 278 TM7 H => Y N/A N/A Gao ZG et al (2000)
aa2ar_human 1.39x39 13 TM1 E => Q N/A N/A Gao ZG et al (2000)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Kim SK et al (2003)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => D N/A N/A Kim SK et al (2003)
aa2ar_human 3.36x36 88 TM3 T => D N/A N/A Jacobson KA et al (2005)
aa2ar_human 3.36x36 88 TM3 T => E N/A N/A Kim SK et al (2003)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Gao ZG et al (2002)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => D N/A N/A Kim SK et al (2003)
aa2ar_human 3.38x38 90 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 4.40x40 119 TM4 T => C N/A N/A Gao ZG et al (2002)
aa2ar_human 151 ECL2 E => A N/A N/A Kim J et al (1996)
aa2ar_human 151 ECL2 E => D N/A N/A Kim J et al (1996)
aa2ar_human 151 ECL2 E => Q N/A N/A Kim J et al (1996)
aa2ar_human 161 ECL2 E => A N/A N/A Kim J et al (1996)
aa2ar_human 169 ECL2 E => A N/A N/A Kim J et al (1996)
aa2ar_human 169 ECL2 E => Q N/A N/A Kim J et al (1996)
aa2ar_human 170 ECL2 D => K N/A N/A Kim J et al (1996)
aa2ar_human 5.34x36 173 TM5 P => R N/A N/A Kim J et al (1996)
aa2ar_human 5.41x42 180 TM5 F => A N/A N/A Kim J et al (1995)
aa2ar_human 5.42x43 181 TM5 N => S N/A N/A Kim J et al (1995)
aa2ar_human 5.43x44 182 TM5 F => A N/A N/A Kim J et al (1995)
aa2ar_human 5.43x44 182 TM5 F => W N/A N/A Kim J et al (1995)
aa2ar_human 5.43x44 182 TM5 F => Y N/A N/A Kim J et al (1995)
aa2ar_human 6.52x52 250 TM6 H => A N/A N/A Gao ZG et al (2002)
aa2ar_human 6.52x52 250 TM6 H => A N/A N/A Kim SK et al (2003)
aa2ar_human 6.52x52 250 TM6 H => A N/A N/A Kim J et al (1995)
aa2ar_human 6.52x52 250 TM6 H => F N/A N/A Kim J et al (1995)
aa2ar_human 6.55x55 253 TM6 N => A N/A N/A Gao ZG et al (2002)
aa2ar_human 6.55x55 253 TM6 N => A N/A N/A Kim SK et al (2003)
aa2ar_human 6.55x55 253 TM6 N => A N/A N/A Kim J et al (1995)
aa2ar_human 6.55x55 253 TM6 N => S N/A N/A Kim J et al (1995)
aa2ar_human 6.56x56 254 TM6 C => A N/A N/A Kim J et al (1995)
aa2ar_human 6.59x59 257 TM6 F => A N/A N/A Kim J et al (1995)
aa2ar_human 6.59x59 257 TM6 F => R N/A N/A Kim J et al (1995)
aa2ar_human 262 ECL3 C => G N/A N/A Scholl DJ et al (2000)
aa2ar_human 262 ECL3 C => G N/A N/A Kim J et al (1996)
aa2ar_human 7.36x35 271 TM7 Y => A N/A N/A Kim J et al (1995)
aa2ar_human 7.39x38 274 TM7 I => A N/A N/A Kim SK et al (2003)
aa2ar_human 7.39x38 274 TM7 I => A N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => A N/A N/A Kim SK et al (2003)
aa2ar_human 7.42x41 277 TM7 S => A N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => C N/A N/A Jiang Q et al (1996)
aa2ar_human 7.42x41 277 TM7 S => D N/A N/A Kim SK et al (2003)
aa2ar_human 7.42x41 277 TM7 S => E N/A N/A Kim SK et al (2003)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.43x42 278 TM7 H => A N/A N/A Kim SK et al (2003)
aa2ar_human 7.43x42 278 TM7 H => A N/A N/A Kim J et al (1995)
aa2ar_human 7.43x42 278 TM7 H => D N/A N/A Kim SK et al (2003)
aa2ar_human 7.43x42 278 TM7 H => E N/A N/A Kim SK et al (2003)
aa2ar_human 7.43x42 278 TM7 H => Q N/A N/A Kim J et al (1995)
aa2ar_human 7.43x42 278 TM7 H => Y N/A N/A Gao ZG et al (2000)
aa2ar_human 7.46x46 281 TM7 S => A N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 7.46x46 281 TM7 S => N N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.39x39 91 TM3 S => A N/A N/A Jiang Q et al (1996)
aa2ar_human 6.55x55 253 TM6 N => Q N/A N/A Kim J et al (1995)
aa2ar_human 6.55x55 253 TM6 N => S N/A N/A Kim J et al (1995)
aa2ar_human 6.55x55 253 TM6 N => A N/A N/A Kim J et al (1995)
aa2ar_human 6.52x52 250 TM6 H => A N/A N/A Kim J et al (1995)
aa2ar_human 5.43x44 182 TM5 F => A N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.46x46 281 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => T N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 7.42x41 277 TM7 S => N N/A N/A Kim J et al (1995)
aa2ar_human 3.37x37 89 TM3 Q => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => H N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => L N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => N N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => R N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => S N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Jiang Q et al (1996)
aa2ar_human 2.61x60 63 TM2 A => H N/A N/A Rosenbaum DM et al (2011)
aa2ar_human 6.55x55 253 TM6 N => A N/A N/A Gao ZG et al (2002)
aa2ar_human 6.52x52 250 TM6 H => A N/A N/A Gao ZG et al (2002)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Gao ZG et al (2002)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Lebon G et al (2011)
aa2ar_human 3.38x38 90 TM3 S => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.55x55 57 TM2 V => A N/A N/A Lebon G et al (2011)
aa2ar_human 154 ECL2 N => A N/A N/A Lebon G et al (2011)
aa2ar_human 3.31x31 83 TM3 F => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.46x46 48 TM2 L => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.63x62 65 TM2 T => A N/A N/A Lebon G et al (2011)
aa2ar_human 154 ECL2 N => A N/A N/A Lebon G et al (2011)
aa2ar_human 6.44x44 242 TM6 F => A N/A N/A Lebon G et al (2011)
aa2ar_human 1.38x38 12 TM1 V => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.48x48 50 TM2 A => L N/A N/A Lebon G et al (2011)
aa2ar_human 2.60x59 62 TM2 F => A N/A N/A Lebon G et al (2011)
aa2ar_human 6.40x40 238 TM6 I => A N/A N/A Lebon G et al (2011)
aa2ar_human 263 ECL3 S => A N/A N/A Lebon G et al (2011)
aa2ar_human 6.38x38 236 TM6 A => L N/A N/A Lebon G et al (2011)
aa2ar_human 3.27x27 79 TM3 F => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.45x45 47 TM2 S => A N/A N/A Lebon G et al (2011)
aa2ar_human 7.47x47 282 TM7 V => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.52x52 54 TM2 A => L N/A N/A Lebon G et al (2011)
aa2ar_human 2.63x62 65 TM2 T => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.52x52 54 TM2 A => L N/A N/A Lebon G et al (2011)
aa2ar_human 3.37x37 89 TM3 Q => A N/A N/A Lebon G et al (2011)
aa2ar_human 2.46x46 48 TM2 L => A N/A N/A Lebon G et al (2011)
aa2ar_human 7.42x41 277 TM7 S => A N/A N/A Dore AS et al (2011)
aa2ar_human 3.55x55 107 TM3 R => A N/A N/A Dore AS et al (2011)
aa2ar_human 2.52x52 54 TM2 A => L N/A N/A Dore AS et al (2011)
aa2ar_human 154 ECL2 N => A N/A N/A Dore AS et al (2011)
aa2ar_human 6.41x41 239 TM6 V => A N/A N/A Dore AS et al (2011)
aa2ar_human 6.37x37 235 TM6 L => A N/A N/A Dore AS et al (2011)
aa2ar_human 4.43x43 122 TM4 K => A N/A N/A Dore AS et al (2011)
aa2ar_human 5.63x63 202 TM5 L => A N/A N/A Dore AS et al (2011)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Dore AS et al (2011)
aa2ar_human 6.51x51 249 TM6 L => A N/A N/A Xu F et al (2011)
aa2ar_human 3.32x32 84 TM3 V => A N/A N/A Xu F et al (2011)
aa2ar_human 3.36x36 88 TM3 T => A N/A N/A Xu F et al (2011)
aa2ar_human 1.39x39 13 TM1 E => Q 15.385↓ IC50 (Binding - Radioligand competition/displacement) CGS21680 IJzerman AP et al (1996) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 1.227↓ IC50 (Binding - Radioligand competition/displacement) CGS 15943 IJzerman AP et al (1996) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 1.13↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE IJzerman AP et al (1996) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 2.331↓ IC50 (Binding - Radioligand saturation) xanthine amine congener IJzerman AP et al (1996) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 8.065↓ EC50 (Functional - cAMP accumulation) CGS21680 IJzerman AP et al (1996) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 1.667↓ K(d) (Binding - Radioligand saturation) ZM-241385 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 2.132↓ k1 (Binding - Radioligand kinetics (association/dissociation)) ZM-241385 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 2.07↓ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM-241385 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 3.03↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 8.929↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 5.495↓ K(i) (Binding - Radioligand competition/displacement) NECA Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 8.13↓ K(i) (Binding - Radioligand competition/displacement) CPA Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 1.0 K(i) (Binding - Radioligand competition/displacement) CGS 15943 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 2.667↑ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 2.105↓ K(i) (Binding - Radioligand competition/displacement) theophylline Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => Q 1.032↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => A 3.981↑ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 1.39x39 13 TM1 E => A 6.329↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 2.50x50 52 TM2 D => A 1.052↑ K(d) (Binding - Radioligand saturation) NECA Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.50x50 52 TM2 D => A 1.314↑ K(d) (Binding - Radioligand saturation) ZM241385 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.50x50 52 TM2 D => A 10.989↓ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.50x50 52 TM2 D => A 14.085↓ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.50x50 52 TM2 D => A 16.949↓ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.50x50 52 TM2 D => A 18.519↓ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.50x50 52 TM2 D => A Abolished effect pEC50 (Functional - cAMP accumulation) CGS21680 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.52x52 54 TM2 A => L 3.03↓ N/A NECA Bertheleme N et al (2013) Jespers W et al (2018)
aa2ar_human 2.52x52 54 TM2 A => L 1.0 K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 2.52x52 54 TM2 A => L 1.767↑ K(i) (Binding - Radioligand competition/displacement) theophylline Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 2.52x52 54 TM2 A => L Abolished effect K(i) (Binding - Radioligand competition/displacement) NECA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 2.52x52 54 TM2 A => L 200.0↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 10.0↓ pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 1.585↓ pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 7.937↓ pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 40.0↓ pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) Chromone1a Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 12.658↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 2.513↓ pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 31.25↓ pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 15.873↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 1.023↑ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 2.64x63 66 TM2 I => A 1.676↑ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => A 3.546↓ pEC50 (Functional - cAMP accumulation) NECA Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => A 1.349↑ pEC50 (Functional - cAMP accumulation) CGS21680 Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => A 1.259↑ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => A 1.545↑ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 2.66x65 68 TM2 T => A 1.047↑ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 2.66x65 68 TM2 T => A 1.053↑ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 23.51x51 71 ECL1 C => A 1.537↑ K(d) (Binding - Radioligand saturation) CGS21680 Naranjo AN et al (2015) Jespers W et al (2018)
aa2ar_human 3.22x22 74 TM3 C => A 1.557↑ K(d) (Binding - Radioligand saturation) CGS21680 Naranjo AN et al (2015) Jespers W et al (2018)
aa2ar_human 3.25x25 77 TM3 C => A 1.35↑ K(d) (Binding - Radioligand saturation) CGS21680 Naranjo AN et al (2015) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 1.333↑ K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 2.016↑ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 1.005↑ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 2.587↑ K(i) (Binding - Radioligand competition/displacement) piclidenoson Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 5.917↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 5.78↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 1.083↓ K(i) (Binding - Radioligand competition/displacement) galangin Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 1.099↑ K(i) (Binding - Radioligand competition/displacement) NIFEDIPINE Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 3.484↓ K(i) (Binding - Radioligand competition/displacement) DPCPX Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 1.46↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL87496 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => L 1.034↑ K(i) (Binding - Radioligand competition/displacement) AMILORIDE Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => D Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => A Abolished effect K(d) (Binding - Radioligand saturation) NECA Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => D Abolished effect K(d) (Binding - Radioligand saturation) NECA Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => D Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.32x32 84 TM3 V => D No effect K(d) (Binding - Radioligand saturation) 3-quinuclidinyl-benzilate Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 62.5↓ pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 200.0↓ pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 12.658↓ pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 40.0↓ pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 62.5↓ pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 20.0↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2030687 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 1000.0↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 500.0↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 7.937↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 12.658↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 7.937↓ pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 12.658↓ pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 12.658↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A N/A pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => R 25.0↓ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => A 100.0↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.33x33 85 TM3 L => R 500.0↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1.222↓ K(d) (Binding - Radioligand saturation) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 1.533↑ K(d) (Binding - Radioligand saturation) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R 2.097↑ K(d) (Binding - Radioligand saturation) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 142.857↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 6.579↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R 76.923↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 90.909↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 10.0↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R 62.5↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 83.333↓ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 40.0↓ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R 142.857↓ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1000.0↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 15.873↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R 166.667↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 6.667↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 5.236↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R 4.167↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 4.587↓ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 1.531↓ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R 2.639↓ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 15.625↓ EC50 (Functional - cAMP accumulation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => S 52.632↓ EC50 (Functional - cAMP accumulation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => R Decreased effect EC50 (Functional - cAMP accumulation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 1.083↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => E 1.254↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D Decreased effect K(i) (Binding - Radioligand competition/displacement) NECA Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => E Abolished effect K(i) (Binding - Radioligand competition/displacement) NECA Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 1.312↑ K(i) (Binding - Radioligand competition/displacement) 5'-Deoxy-5'-aminoadenosine Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => E 1.085↑ K(i) (Binding - Radioligand competition/displacement) 5'-Deoxy-5'-aminoadenosine Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 3.722↑ K(i) (Binding - Radioligand competition/displacement) CID 85129620 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => E 1.175↑ K(i) (Binding - Radioligand competition/displacement) CID 85129620 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 12.154↑ K(i) (Binding - Radioligand competition/displacement) 522607-99-4 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => E 1.234↑ K(i) (Binding - Radioligand competition/displacement) 522607-99-4 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 10.477↑ K(i) (Binding - Radioligand competition/displacement) Cid13307390 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => E 1.236↓ K(i) (Binding - Radioligand competition/displacement) Cid13307390 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 1.751↓ K(d) (Binding - Radioligand saturation) ZM241385 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D Abolished effect K(i) (Binding - Radioligand competition/displacement) CHEMBL277076 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 1.083↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018681 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 1.259↓ K(i) (Binding - Radioligand competition/displacement) NONAME Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 2.985↓ K(i) (Binding - Radioligand competition/displacement) CID 75022550 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 1.288↑ K(i) (Binding - Radioligand competition/displacement) Cid76018682 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018683 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018684 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 1.835↓ K(i) (Binding - Radioligand competition/displacement) CAS35788-28-4 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018685 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D Abolished effect K(i) (Binding - Radioligand competition/displacement) Oprea1_724488 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018686 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018687 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) NCGC00015640-02 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid44280242 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid22948626 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018688 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 3.597↓ EC50 (Functional - cAMP accumulation) NONAME Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => D 2.174↓ EC50 (Functional - cAMP accumulation) Cid76018686 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1.259↑ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1000.0↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1.097↑ K(d) (Binding - Radioligand saturation) ZM241385 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A Abolished effect pK(i) (Binding - Radioligand competition/displacement) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1.585↓ pK(i) (Binding - Radioligand competition/displacement) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A Abolished effect N/A NECA Bertheleme N et al (2013) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 200.0↓ K(i) (Binding - Radioligand competition/displacement) NECA Bertheleme N et al (2013) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 7.519↓ K(i) (Binding - Radioligand competition/displacement) adenosine Bertheleme N et al (2013) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 83.333↓ EC50 (Functional - Other) adenosine Bertheleme N et al (2013) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1.0 K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 1.767↑ K(i) (Binding - Radioligand competition/displacement) theophylline Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A Abolished effect K(i) (Binding - Radioligand competition/displacement) NECA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 3.36x36 88 TM3 T => A 200.0↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 670.732↑ K(i) (Binding - Radioligand competition/displacement) CID 75022550 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 50.6↑ K(i) (Binding - Radioligand competition/displacement) CAS35788-28-4 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 100.0↑ EC50 (Functional - cAMP accumulation) Cid76018686 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 2.665↑ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 4.103↑ EC50 (Functional - cAMP accumulation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 7.52↑ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 2.4↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 2.4↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 4.286↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 14.267↑ K(i) (Binding - Radioligand competition/displacement) NECA Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 14.267↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL277076 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 14.526↑ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 4.333↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 3.956↑ EC50 (Functional - cAMP accumulation) CGS 24012 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 15.292↑ EC50 (Functional - cAMP accumulation) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 135.514↑ K(i) (Binding - Radioligand competition/displacement) piclidenoson Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 12.806↑ K(i) (Binding - Radioligand competition/displacement) Cid13307390 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 1.916↓ K(d) (Binding - Radioligand saturation) ZM241385 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 161.961↑ EC50 (Functional - cAMP accumulation) NONAME Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 10.469↑ K(i) (Binding - Radioligand competition/displacement) CID 85129620 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 4.627↑ K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 4.627↑ K(d) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 6.87↑ K(i) (Binding - Radioligand competition/displacement) Cid76018682 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 5.236↑ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 10.455↑ K(i) (Binding - Radioligand competition/displacement) R-PIA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => L 1.148↓ K(d) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 32.282↑ K(i) (Binding - Radioligand competition/displacement) ADAC Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => H 1.511↓ K(d) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => R 1.639↓ K(d) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 10.269↑ K(i) (Binding - Radioligand competition/displacement) 5'-Deoxy-5'-aminoadenosine Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 1.362↑ K(i) (Binding - Radioligand competition/displacement) 522607-99-4 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => S 3.012↓ K(d) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => N 3.185↓ K(d) (Binding - Radioligand competition/displacement) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => A 6.459↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL87496 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 10.528↑ K(i) (Binding - Radioligand competition/displacement) Oprea1_724488 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D 5.834↑ K(i) (Binding - Radioligand competition/displacement) NONAME Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018681 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018683 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018684 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018685 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018686 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018687 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D No effect K(i) (Binding - Radioligand competition/displacement) NCGC00015640-02 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D No effect K(i) (Binding - Radioligand competition/displacement) Cid44280242 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D No effect K(i) (Binding - Radioligand competition/displacement) Cid22948626 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.37x37 89 TM3 Q => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018688 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 1.925↑ K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 5.155↑ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 4.678↑ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 3.929↑ K(i) (Binding - Radioligand competition/displacement) R-PIA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 5.541↑ K(i) (Binding - Radioligand competition/displacement) piclidenoson Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 1.97↑ K(i) (Binding - Radioligand competition/displacement) ADAC Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 1.233↑ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 2.108↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 1.905↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 1.691↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL87496 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.38x38 90 TM3 S => A 1.458↑ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.927↓ K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 2.242↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.287↓ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.05↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.412↓ K(i) (Binding - Radioligand competition/displacement) piclidenoson Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.901↓ K(i) (Binding - Radioligand competition/displacement) ADAC Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.244↓ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.0 K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 2.079↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 2.188↓ K(i) (Binding - Radioligand competition/displacement) CHEMBL87496 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 2.075↓ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 3.185↓ K(d) (Binding - Radioligand saturation) NECA Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.522↓ K(d) (Binding - Radioligand saturation) ZM241385 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.231↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.087↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.302↓ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A 1.085↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 3.39x39 91 TM3 S => A No effect pEC50 (Functional - cAMP accumulation) CGS21680 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 4.43x43 122 TM4 K => A 1.0 K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 4.43x43 122 TM4 K => A 1.767↑ K(i) (Binding - Radioligand competition/displacement) theophylline Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 4.43x43 122 TM4 K => A Abolished effect K(i) (Binding - Radioligand competition/displacement) NECA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 4.43x43 122 TM4 K => A 200.0↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 146 ECL2 C => A 1.828↑ K(d) (Binding - Radioligand saturation) CGS21680 Naranjo AN et al (2015) Jespers W et al (2018)
aa2ar_human 148 ECL2 Q => A 1.122↓ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 148 ECL2 Q => A 1.244↓ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 150 ECL2 K => A 1.099↓ K(d) (Binding - Radioligand saturation) ZM241385 Moss SM et al (2014) Jespers W et al (2018)
aa2ar_human 151 ECL2 E => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 151 ECL2 E => Q Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 151 ECL2 E => D Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 151 ECL2 E => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 151 ECL2 E => Q Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 151 ECL2 E => D Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 153 ECL2 K => A 1.231↑ K(d) (Binding - Radioligand saturation) ZM241385 Moss SM et al (2014) Jespers W et al (2018)
aa2ar_human 153 ECL2 K => A 1.202↑ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 153 ECL2 K => A 1.266↑ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 154 ECL2 N => Q No effect K(d) (Binding - Radioligand saturation) ZM-241385 Fraser NJ et al (2006) Jespers W et al (2018)
aa2ar_human 154 ECL2 N => Q No effect K(i) (Binding - Radioligand competition/displacement) ZM-241385 Fraser NJ et al (2006) Jespers W et al (2018)
aa2ar_human 154 ECL2 N => Q No effect K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Fraser NJ et al (2006) Jespers W et al (2018)
aa2ar_human 154 ECL2 N => Q Increased effect K(i) (Binding - Radioligand competition/displacement) CHEMBL277076 Fraser NJ et al (2006) Jespers W et al (2018)
aa2ar_human 154 ECL2 N => Q No effect K(i) (Binding - Radioligand competition/displacement) theophylline Fraser NJ et al (2006) Jespers W et al (2018)
aa2ar_human 156 ECL2 S => A 1.413↑ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 156 ECL2 S => A 1.075↓ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 157 ECL2 Q => A 1.585↑ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 157 ECL2 Q => A 1.062↑ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 159 ECL2 C => A 1.898↑ K(d) (Binding - Radioligand saturation) CGS21680 Naranjo AN et al (2015) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 1.869↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 1.534↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 1.686↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 1.672↓ K(i) (Binding - Radioligand competition/displacement) (R)-PIA Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 1.053↑ K(i) (Binding - Radioligand competition/displacement) piclidenoson Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 2.096↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 5.958↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 161 ECL2 E => A 1.03↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 45.50x50 166 ECL2 C => A 1.467↑ K(d) (Binding - Radioligand saturation) CGS21680 Naranjo AN et al (2015) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.0 pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 10.0↓ pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.585↓ pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.0 pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2030687 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 2.513↓ pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 2.513↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 1.995↑ pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 25.0↓ pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => Y 8.13↓ K(d) (Binding - Radioligand saturation) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => W 4.0↓ K(d) (Binding - Radioligand saturation) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => A Abolished effect K(d) (Binding - Radioligand saturation) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => Y 2.294↓ K(d) (Binding - Other) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => W 1.499↓ K(d) (Binding - Other) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => A Abolished effect K(d) (Binding - Other) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => Y 12.658↓ K(i) (Binding - Radioligand competition/displacement) NECA Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => W 2.41↑ K(i) (Binding - Radioligand competition/displacement) NECA Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => Y 25.0↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => W 1.495↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => Y 1.09↑ EC50 (Functional - cAMP accumulation) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => W 1.019↑ EC50 (Functional - cAMP accumulation) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => A 1.307↑ EC50 (Functional - cAMP accumulation) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => A 500.0↓ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => D Abolished effect pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => A 500.0↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 45.52x52 168 ECL2 F => D Abolished effect pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 2.558↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 6.579↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 22.407↑ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 4.661↑ K(i) (Binding - Radioligand competition/displacement) (R)-PIA Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 8.539↑ K(i) (Binding - Radioligand competition/displacement) piclidenoson Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 22.222↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 1.321↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 1.647↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A 3.162↑ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A 1.259↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A 29.412↓ pIC50 (Functional - Ca2+ accumulation) ZM241385 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A 15.152↓ pEC50 (Functional - cAMP accumulation) NECA Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A 1.585↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A Abolished effect pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 2.342↓ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => A Abolished effect k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 169 ECL2 E => Q 62.5↓ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 170 ECL2 D => K No effect (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 170 ECL2 D => K No effect (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 5.34x36 173 TM5 P => R No effect (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 5.34x36 173 TM5 P => R No effect (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 7.937↓ pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.585↓ pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A Decreased effect pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A Decreased effect pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL2030687 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.0 pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A Decreased effect pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.585↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A Decreased effect pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.0 pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.0 pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A Decreased effect pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 3.162↑ pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 7.519↓ K(d) (Binding - Radioligand saturation) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 4.329↓ K(d) (Binding - Other) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.424↑ K(i) (Binding - Radioligand competition/displacement) NECA Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 6.849↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 5.38x40 177 TM5 M => A 1.112↑ EC50 (Functional - cAMP accumulation) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 5.41x42 180 TM5 F => A 1.437↑ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.41x42 180 TM5 F => A 2.346↑ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.41x42 180 TM5 F => A 2.309↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.41x42 180 TM5 F => A 14.085↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.41x42 180 TM5 F => A 1.357↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.41x42 180 TM5 F => A 1.429↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.41x42 180 TM5 F => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 7.937↓ pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 15.873↓ pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 2.513↓ pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 3.981↑ pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 2.513↓ pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2030687 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 2.513↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 1.585↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 20.0↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 10.0↓ pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => S 1.143↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => S 8.85↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => S 4.016↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => S 1.213↑ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => S 2.347↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => S 2.058↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 1.709↓ K(d) (Binding - Radioligand saturation) ZM241385 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 2.301↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL277076 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 1.867↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018681 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 3.956↑ K(i) (Binding - Radioligand competition/displacement) NONAME Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 9.322↑ K(i) (Binding - Radioligand competition/displacement) CID 75022550 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 93.509↑ K(i) (Binding - Radioligand competition/displacement) Cid13307390 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 17.923↑ K(i) (Binding - Radioligand competition/displacement) Cid76018682 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018683 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018684 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 6.289↓ K(i) (Binding - Radioligand competition/displacement) CAS35788-28-4 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018685 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 1.34↓ K(i) (Binding - Radioligand competition/displacement) Oprea1_724488 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018686 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) Cid76018687 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D No effect K(i) (Binding - Radioligand competition/displacement) NCGC00015640-02 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D No effect K(i) (Binding - Radioligand competition/displacement) Cid44280242 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D No effect K(i) (Binding - Radioligand competition/displacement) Cid22948626 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D No effect K(i) (Binding - Radioligand competition/displacement) Cid76018688 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 6.883↑ EC50 (Functional - cAMP accumulation) NONAME Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.42x43 181 TM5 N => D 111.538↑ EC50 (Functional - cAMP accumulation) Cid76018686 Jacobson KA et al (2005) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => Y 2.625↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => W 3.04↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => Y 12.5↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => W 5.102↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => Y 7.042↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => W 3.096↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => Y 8.547↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => W 7.246↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => Y 8.772↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => W 5.025↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => Y 1.901↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => W 1.019↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => Y 2.217↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => W 1.057↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 5.43x44 182 TM5 F => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.41x41 239 TM6 V => A 111.111↓ N/A NECA Bertheleme N et al (2013) Jespers W et al (2018)
aa2ar_human 6.41x41 239 TM6 V => A 1.0 K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 6.41x41 239 TM6 V => A 1.767↑ K(i) (Binding - Radioligand competition/displacement) theophylline Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 6.41x41 239 TM6 V => A Abolished effect K(i) (Binding - Radioligand competition/displacement) NECA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 6.41x41 239 TM6 V => A 200.0↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Magnani F et al (2008) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 3.162↑ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => Y 79.433↑ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 40.0↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => Y 3.162↑ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 23.81↓ K(d) (Binding - Radioligand saturation) NECA Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 5.051↓ K(d) (Binding - Radioligand saturation) ZM241385 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 5.926↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 5.814↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 24.231↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 24.722↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 5.0↓ pEC50 (Functional - cAMP accumulation) CGS21680 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 10.309↓ % (Binding - Radioligand competition/displacement) 12a Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 23.81↓ % (Binding - Radioligand competition/displacement) 12b Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 2.874↓ % (Binding - Radioligand competition/displacement) 12c Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 7.463↓ % (Binding - Radioligand competition/displacement) 12d Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 13.889↓ % (Binding - Radioligand competition/displacement) 12e Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 11.765↓ % (Binding - Radioligand competition/displacement) 12f Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 7.576↓ % (Binding - Radioligand competition/displacement) 12g Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A N/A % (Binding - Radioligand competition/displacement) CHEMBL3819703 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 7.576↓ % (Binding - Radioligand competition/displacement) CHEMBL3819730 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 28.571↓ % (Binding - Radioligand competition/displacement) 12j Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 34.483↓ % (Binding - Radioligand competition/displacement) CHEMBL3819709 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 7.692↓ % (Binding - Radioligand competition/displacement) CHEMBL3819710 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 19.608↓ % (Binding - Radioligand competition/displacement) 12m Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 19.231↓ % (Binding - Radioligand competition/displacement) 12n Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 18.868↓ % (Binding - Radioligand competition/displacement) 12o Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 12.048↓ % (Binding - Radioligand competition/displacement) 12p Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 6.452↓ % (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 16.667↓ % (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.261↑ % (Binding - Radioligand competition/displacement) CID11277660 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.812↓ % (Binding - Radioligand competition/displacement) CID57403241 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.372↓ % (Binding - Radioligand competition/displacement) CID57396267 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 3.817↓ % (Binding - Radioligand competition/displacement) CID57392705 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.02↑ % (Binding - Radioligand competition/displacement) CID57392707 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 3.663↓ % (Binding - Radioligand competition/displacement) CID57399649 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.543↓ % (Binding - Radioligand competition/displacement) CID57403156 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.192↓ % (Binding - Radioligand competition/displacement) CID57399651 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 2.0↓ % (Binding - Radioligand competition/displacement) CID57394421 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 50.0↓ % (Binding - Radioligand competition/displacement) CID44574895 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 6.667↓ % (Binding - Radioligand competition/displacement) compound_13 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.603↓ % (Binding - Radioligand competition/displacement) CID57390905 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 1.385↓ % (Binding - Radioligand competition/displacement) CID57397997 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 2.398↓ % (Binding - Radioligand competition/displacement) CID57390907 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 4.545↓ % (Binding - Radioligand competition/displacement) CID57394423 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 2.66↓ % (Binding - Radioligand competition/displacement) CID57401407 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 18.889↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 36.667↑ IC50 (Binding - Radioligand competition/displacement) CHEMBL3819703 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 32.4↑ IC50 (Binding - Radioligand competition/displacement) CHEMBL3819730 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 80.0↑ IC50 (Binding - Radioligand competition/displacement) CHEMBL3819709 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 68.0↑ IC50 (Binding - Radioligand competition/displacement) CHEMBL3819710 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 20.0↑ RT (Binding - Radioligand kinetics (association/dissociation)) 5-(N,N-hexamethylene)-amiloride Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 22.0↑ RT (Binding - Radioligand kinetics (association/dissociation)) CHEMBL3819703 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 52.5↑ RT (Binding - Radioligand kinetics (association/dissociation)) CHEMBL3819730 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 50.833↑ RT (Binding - Radioligand kinetics (association/dissociation)) CHEMBL3819709 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 30.769↑ RT (Binding - Radioligand kinetics (association/dissociation)) CHEMBL3819710 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.48x48 246 TM6 W => A 21.786↑ RT (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Massink A et al (2016) Jespers W et al (2018)
aa2ar_human 6.51x51 249 TM6 L => A Abolished effect K(d) (Binding - Radioligand saturation) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 6.51x51 249 TM6 L => A Abolished effect K(d) (Binding - Other) ZM241385 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 6.51x51 249 TM6 L => A 1.172↑ EC50 (Functional - cAMP accumulation) CGS21680 Jaakola VP et al (2010) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => F 1.507↑ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => Y 1.456↑ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => F 14.085↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => Y 55.556↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => F 6.757↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => Y 12.346↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => F 2.105↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => Y 2.203↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => F 25.0↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => Y 30.303↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => F 2.545↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => Y 1.202↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => F 1.048↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => Y 1.199↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 4.789↑ K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 1.061↑ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 4.122↑ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 11.562↑ K(i) (Binding - Radioligand competition/displacement) piclidenoson Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 3.215↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 1.976↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 1.976↓ K(i) (Binding - Radioligand competition/displacement) galangin Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 1.099↑ K(i) (Binding - Radioligand competition/displacement) NIFEDIPINE Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 1.287↓ K(i) (Binding - Radioligand competition/displacement) DPCPX Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 1.952↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL87496 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.52x52 250 TM6 H => N 3.659↑ K(i) (Binding - Radioligand competition/displacement) AMILORIDE Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) CHEMBL2030687 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => S Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => Q Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => S Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => Q Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A Abolished effect pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 6.55x55 253 TM6 N => A 166.667↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 6.56x56 254 TM6 C => A 1.092↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.56x56 254 TM6 C => A 2.45↑ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.56x56 254 TM6 C => A 1.093↑ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.56x56 254 TM6 C => A 1.919↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.56x56 254 TM6 C => A 1.168↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.56x56 254 TM6 C => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.58x58 256 TM6 T => A 2.513↓ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 6.58x58 256 TM6 T => A 16.667↓ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 6.59x59 257 TM6 F => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.59x59 257 TM6 F => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 6.59x59 257 TM6 F => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 262 ECL3 C => G No effect (Binding - Radioligand saturation) CGS21680 Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 262 ECL3 C => G No effect (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1996) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 2.512↑ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 3.984↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 7.407↓ pEC50 (Functional - cAMP accumulation) NECA Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 5.618↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 1.381↓ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 18.868↓ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 1.276↑ % (Binding - Radioligand saturation) CHEMBL184061 Segala E et al (2016) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 1.0 % (Binding - Radioligand saturation) CHEMBL3937413 Segala E et al (2016) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => A 1.01↑ % (Binding - Radioligand saturation) ZM241385 Segala E et al (2016) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => Q 1.342↑ % (Binding - Radioligand saturation) CHEMBL184061 Segala E et al (2016) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => Q 1.0 % (Binding - Radioligand saturation) CHEMBL3937413 Segala E et al (2016) Jespers W et al (2018)
aa2ar_human 264 ECL3 H => Q 1.082↓ % (Binding - Radioligand saturation) ZM241385 Segala E et al (2016) Jespers W et al (2018)
aa2ar_human 7.32x31 267 TM7 L => A 1.739↓ pEC50 (Functional - cAMP accumulation) NECA Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 7.32x31 267 TM7 L => A 24.547↑ pEC50 (Functional - cAMP accumulation) CGS21680 Lebon G et al (2015) Jespers W et al (2018)
aa2ar_human 7.32x31 267 TM7 L => A 1.122↓ pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 7.32x31 267 TM7 L => A 2.333↑ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 7.937↓ pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.0 pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.0 pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 5.0↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2030687 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.0 pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 3.165↓ pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 6.329↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.996↓ pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.585↓ pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 1.259↓ pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 25.0↓ pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A 12.658↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A Abolished effect pK(i) (Binding - Radioligand competition/displacement) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 7.36x35 271 TM7 Y => A Abolished effect k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM241385 Guo D et al (2016) Jespers W et al (2018)
aa2ar_human 7.39x38 274 TM7 I => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.39x38 274 TM7 I => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.39x38 274 TM7 I => A 33.333↓ EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 2.513↓ pK(d) (Biing - Surface plasmon resonance) ZM-241385 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 7.937↓ pK(d) (Biing - Surface plasmon resonance) preladenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 5.012↑ pK(d) (Biing - Surface plasmon resonance) istradefylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.995↑ pK(d) (Biing - Surface plasmon resonance) xanthine amine congener Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 5.012↑ pK(d) (Biing - Surface plasmon resonance) caffeine Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.0 pK(d) (Biing - Surface plasmon resonance) theophylline Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.995↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL2030687 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.995↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL3133072 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.585↑ pK(d) (Biing - Surface plasmon resonance) Chromone1c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.259↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL1330311 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.0 pK(d) (Biing - Surface plasmon resonance) CHEMBL3133071 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 3.984↓ pK(d) (Biing - Surface plasmon resonance) NOTDISCLOSED Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 10.0↓ pK(d) (Biing - Surface plasmon resonance) CHEMBL1800358 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 10.0↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL3260728 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.995↑ pK(d) (Biing - Surface plasmon resonance) Triazine3b Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 6.31↑ pK(d) (Biing - Surface plasmon resonance) Triazine3c Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 7.943↑ pK(d) (Biing - Surface plasmon resonance) compound 4g [PMID: 22220592] Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 15.849↑ pK(d) (Biing - Surface plasmon resonance) imaradenant Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 25.119↑ pK(d) (Biing - Surface plasmon resonance) Triazine3f Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 5.012↑ pK(d) (Biing - Surface plasmon resonance) Triazine3g Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 6.31↑ pK(d) (Biing - Surface plasmon resonance) CHEMBL2024119 Zhukov A et al (2011) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => N 1.152↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => T 1.088↓ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => N 1.453↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => T 1.323↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => N 1.274↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => T 1.25↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => N 2.16↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => T 2.0↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => N 1.984↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => T 1.678↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => N 1.267↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => T 1.208↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => N 1.053↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => T 1.043↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.403↑ K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1000.0↓ K(i) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 333.333↓ K(i) (Binding - Radioligand saturation) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 111.111↓ K(i) (Binding - Radioligand saturation) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 66.667↓ K(i) (Binding - Radioligand saturation) piclidenoson Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 500.0↓ K(i) (Binding - Radioligand saturation) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 43.478↓ K(i) (Binding - Radioligand saturation) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.183↑ K(i) (Binding - Radioligand saturation) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 3.027↑ K(i) (Binding - Radioligand saturation) DPCPX Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 71.429↓ EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 1.2↓ K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 3.846↓ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 4.673↓ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 5.319↓ K(i) (Binding - Radioligand competition/displacement) R-PIA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 4.032↓ K(i) (Binding - Radioligand competition/displacement) piclidenoson Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 2.688↓ K(i) (Binding - Radioligand competition/displacement) ADAC Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 2.538↓ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 1.275↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 1.182↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 3.079↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL87496 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => C 2.571↓ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => E 1.19↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => E 1.364↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => E 1.131↓ K(i) (Binding - Radioligand competition/displacement) 5'-Deoxy-5'-aminoadenosine Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => E 1.314↓ K(i) (Binding - Radioligand competition/displacement) CID 85129620 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => E 1.179↑ K(i) (Binding - Radioligand competition/displacement) 522607-99-4 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => E 1.124↑ K(i) (Binding - Radioligand competition/displacement) Cid13307390 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 2.512↑ pEC50 (Functional - cAMP accumulation) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 125.0↓ pEC50 (Functional - cAMP accumulation) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 1.172↑ K(d) (Binding - Radioligand saturation) ZM241385 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A Abolished effect pK(i) (Binding - Radioligand competition/displacement) LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A 5.012↑ pK(i) (Binding - Radioligand competition/displacement) CGS21680 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 7.42x41 277 TM7 S => A N/A N/A LUF-5834 Lane JR et al (2012) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Q Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => F Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Q Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => F Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => A 333.333↓ EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => K Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => N Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => K Abolished effect K(d) (Binding - Radioligand saturation) NECA Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => N Abolished effect K(d) (Binding - Radioligand saturation) NECA Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => K Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => N Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Jiang Q et al (1997) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 2.387↓ K(d) (Binding - Radioligand saturation) ZM-241385 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 1.667↓ k1 (Binding - Radioligand kinetics (association/dissociation)) ZM-241385 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 1.757↓ k-1 (Binding - Radioligand kinetics (association/dissociation)) ZM-241385 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 9.709↓ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 71.429↓ K(i) (Binding - Radioligand competition/displacement) CGS21680 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 250.0↓ K(i) (Binding - Radioligand competition/displacement) NECA Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 13.889↓ K(i) (Binding - Radioligand competition/displacement) CPA Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 3.003↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 2.667↑ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 20.833↓ K(i) (Binding - Radioligand competition/displacement) theophylline Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => Y 2.033↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Gao ZG et al (2000) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => D 2.049↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => E 1.615↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => D 1.12↑ K(i) (Binding - Radioligand competition/displacement) NECA Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => E 1.149↓ K(i) (Binding - Radioligand competition/displacement) NECA Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => D 1.299↓ K(i) (Binding - Radioligand competition/displacement) CID 85129620 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => E 1.047↑ K(i) (Binding - Radioligand competition/displacement) CID 85129620 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => D 1.339↑ K(i) (Binding - Radioligand competition/displacement) 522607-99-4 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => E 1.411↑ K(i) (Binding - Radioligand competition/displacement) 522607-99-4 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => D 2.625↓ K(i) (Binding - Radioligand competition/displacement) Cid13307390 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.43x42 278 TM7 H => E 1.562↓ K(i) (Binding - Radioligand competition/displacement) Cid13307390 Kim SK et al (2003) Jespers W et al (2018)
aa2ar_human 7.45x45 280 TM7 N => A 9.259↓ K(d) (Binding - Radioligand saturation) NECA Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.45x45 280 TM7 N => A 1.825↓ K(d) (Binding - Radioligand saturation) ZM241385 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.45x45 280 TM7 N => A 1.6↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.45x45 280 TM7 N => A 1.042↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.45x45 280 TM7 N => A 3.15↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.45x45 280 TM7 N => A 3.56↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.45x45 280 TM7 N => A 1.0 pEC50 (Functional - cAMP accumulation) CGS21680 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => T 1.269↑ K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => A Abolished effect K(d) (Binding - Radioligand saturation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => T 11.095↑ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => T 3.031↑ K(i) (Binding - Radioligand competition/displacement) CGS 24012 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => T 3.015↑ K(i) (Binding - Radioligand competition/displacement) NECA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => T 10.426↑ K(i) (Binding - Radioligand competition/displacement) R-PIA Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => T 1.546↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => T 3.653↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => A Abolished effect K(d) (Binding - Radioligand saturation) xanthine amine congener Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => A Abolished effect EC50 (Functional - cAMP accumulation) CGS21680 Kim J et al (1995) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 2.52↑ K(d) (Binding - Radioligand saturation) CGS21680 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 13.459↑ K(i) (Binding - Radioligand competition/displacement) 2-chloroadenosine Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 6.133↑ K(i) (Binding - Radioligand competition/displacement) NECA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 16.989↑ K(i) (Binding - Radioligand competition/displacement) R-PIA Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 8.116↑ K(i) (Binding - Radioligand competition/displacement) piclidenoson Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 8.526↑ K(i) (Binding - Radioligand competition/displacement) ADAC Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 4.237↓ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 2.618↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 9.434↓ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 3.506↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL87496 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.46x46 281 TM7 S => N 3.676↓ K(i) (Binding - Radioligand competition/displacement) ZM241385 Jiang Q et al (1996) Jespers W et al (2018)
aa2ar_human 7.49x49 284 TM7 N => A 2.924↓ K(d) (Binding - Radioligand saturation) NECA Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.49x49 284 TM7 N => A 1.522↓ K(d) (Binding - Radioligand saturation) ZM241385 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.49x49 284 TM7 N => A 2.712↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.49x49 284 TM7 N => A 2.5↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.49x49 284 TM7 N => A 3.938↑ IC50 (Binding - Radioligand competition/displacement) AMILORIDE Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.49x49 284 TM7 N => A 2.697↑ IC50 (Binding - Radioligand competition/displacement) 5-(N,N-hexamethylene)-amiloride Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 7.49x49 284 TM7 N => A Abolished effect pEC50 (Functional - cAMP accumulation) CGS21680 Massink A et al (2015) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 2.89↑ K(i) (Binding - Radioligand competition/displacement) ZM241385 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 1.58↑ K(i) (Binding - Radioligand competition/displacement) ZM241385 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 1.27↑ K(i) (Binding - Radioligand competition/displacement) ZM241385 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 4.03↑ K(i) (Binding - Radioligand competition/displacement) ZM241385 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 2.44↑ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 1.67↑ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 1.235↓ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 3.8↑ K(i) (Binding - Radioligand competition/displacement) SCH 58261 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 3.85↑ K(i) (Binding - Radioligand competition/displacement) SCH442416 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 7.3↑ K(i) (Binding - Radioligand competition/displacement) SCH442416 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 1.429↓ K(i) (Binding - Radioligand competition/displacement) SCH442416 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 6.68↑ K(i) (Binding - Radioligand competition/displacement) SCH442416 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 2.88↑ K(i) (Binding - Radioligand competition/displacement) istradefylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 2.79↑ K(i) (Binding - Radioligand competition/displacement) istradefylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 1.33↑ K(i) (Binding - Radioligand competition/displacement) istradefylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 1.51↑ K(i) (Binding - Radioligand competition/displacement) istradefylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 1.35↑ K(i) (Binding - Radioligand competition/displacement) PSB36 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 1.19↓ K(i) (Binding - Radioligand competition/displacement) PSB36 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 1.19↓ K(i) (Binding - Radioligand competition/displacement) PSB36 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 5.0↓ K(i) (Binding - Radioligand competition/displacement) PSB36 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 1.48↑ K(i) (Binding - Radioligand competition/displacement) DPCPX Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 1.51↑ K(i) (Binding - Radioligand competition/displacement) DPCPX Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 1.37↓ K(i) (Binding - Radioligand competition/displacement) DPCPX Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 5.556↓ K(i) (Binding - Radioligand competition/displacement) DPCPX Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 3.11↑ K(i) (Binding - Radioligand competition/displacement) rolofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 1.87↑ K(i) (Binding - Radioligand competition/displacement) rolofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 2.15↑ K(i) (Binding - Radioligand competition/displacement) rolofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 5.0↓ K(i) (Binding - Radioligand competition/displacement) rolofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 2.222↓ K(i) (Binding - Radioligand competition/displacement) derenofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 4.78↑ K(i) (Binding - Radioligand competition/displacement) derenofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 1.02↓ K(i) (Binding - Radioligand competition/displacement) derenofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 1.1↑ K(i) (Binding - Radioligand competition/displacement) derenofylline Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 3.61↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 3.9↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 2.32↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 1.38↑ K(i) (Binding - Radioligand competition/displacement) xanthine amine congener Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.57x56 59 TM2 A => V 2.11↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 2.65x64 67 TM2 S => N 1.67↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 45.51x51 167 ECL2 L => E 2.0↓ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 1.47↑ K(i) (Binding - Radioligand competition/displacement) CGS 15943 Cheng RKY et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 6.31↑ pK(i) (Binding - Radioligand competition/displacement) DPCPX Glukhova A et al (2017) Jespers W et al (2018)
aa2ar_human 7.35x34 270 TM7 M => T 7.937↓ pK(i) (Binding - Radioligand competition/displacement) SCH 58261 Glukhova A et al (2017) Jespers W et al (2018)
aa2ar_human 153 ECL2 K => A 1.202↓ pK(i) (Binding - Radioligand competition/displacement) SCH 58261 Yang X et al (2017) Jespers W et al (2018)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 S N L Q ICL1ECL1 F C A ECL1ICL2 P L R Y N G L V ICL2ECL2 W N N C G Q P K E G K N H S Q G C G E G Q V A C L F E D V V ECL2ICL3 Q P L P G ICL3ECL3 P D C S H A ECL3C-term K A A G T S A R V L A A H G S D G E Q V S L R L N G H P P G V W A N G S A P H P E R R P N G Y A L G L V S G G S A Q E S Q G N T G L P D V E L L S H E L K G V C P E P P G L D D P L A Q D G A G V S C-term M P I M G S S V Y I T V E L A I A V L A I L G N V L V C W A V W L N N V T N Y F V V S L A A A D I A V G V L A I P F A I T I S T G A C H G C L F I A C F V L V L T Q S S I F S L L A I A I D R Y I A I R I T G T R A K G I I A I C W V L S F A I G L T P M L G P M N Y M V Y F N F F A C V L V P L L L M L G V Y L R I F L A A R R Q L K Q M E S E R A R S T L Q K E V H A A K S L A I I V G L F A L C W L P L H I I N C F T F F C P L W L M Y L A I V L S H T N S V V N P F I Y A Y R I R E F R K H V L P F F R Q T I I R S R Q Q E
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
V N G L I A L V A I A L E V T I Y V S S 1 V S L A A A D I A V G L V A I P F A I T I 2 A L L S F I S S Q T L V L V F C A I F L 3 A K G I I A I C W V L S F A I G L T P M 4 Y V G L M L L L P V L V C A F F N F Y V M Y 5 A I I V G L F A L C W L P L H I I N C F 6 F P N V V S N T H S L V I A L Y M L W 7
Download: PNG | SVG




Residue Table


GPCRdb(A)
GPCRdb(A)
A2A receptor
TM1
1x38 1.38x38 V12
1x39 1.39x39 E13
TM2
2x45 2.45x45 S47
2x46 2.46x46 L48
2x48 2.48x48 A50
2x50 2.50x50 D52
2x52 2.52x52 A54
2x55 2.55x55 V57
2x56 2.57x56 A59
2x59 2.60x59 F62
2x60 2.61x60 A63
2x62 2.63x62 T65
2x63 2.64x63 I66
2x64 2.65x64 S67
2x65 2.66x65 T68
TM3
3x22 3.22x22 C74
3x23 3.23x23 H75
3x25 3.25x25 C77
3x27 3.27x27 F79
3x31 3.31x31 F83
3x32 3.32x32 V84
3x33 3.33x33 L85
3x36 3.36x36 T88
3x37 3.37x37 Q89
3x38 3.38x38 S90
3x39 3.39x39 S91
3x55 3.55x55 R107
TM4
4x39 4.39x39 G118
4x40 4.40x40 T119
4x43 4.43x43 K122
4x44 4.44x44 G123
TM5
5x36 5.34x36 P173
5x40 5.38x40 M177
5x42 5.41x42 F180
5x43 5.42x43 N181
5x44 5.43x44 F182
5x46 5.45x46 A184
5x60 5.60x60 R199
5x63 5.63x63 L202
5x64 5.64x64 A203
5x65 5.65x65 A204
5x69 5.69x69 L208
5x71 5.71x71 Q210
5x74 5.74x74 S213
TM6
6x21 6.21x21 E219
6x22 6.22x22 R220
6x25 6.25x25 S223
6x26 6.26x26 T224
6x28 6.28x28 Q226
6x29 6.29x29 K227
6x32 6.32x32 H230
6x33 6.33x33 A231
6x37 6.37x37 L235
6x38 6.38x38 A236
6x40 6.40x40 I238
6x41 6.41x41 V239
6x43 6.43x43 L241
6x44 6.44x44 F242
6x48 6.48x48 W246
6x51 6.51x51 L249
6x52 6.52x52 H250
6x55 6.55x55 N253
6x56 6.56x56 C254
6x58 6.58x58 T256
6x59 6.59x59 F257
TM7
7x31 7.32x31 L267
7x34 7.35x34 M270
7x35 7.36x35 Y271
7x36 7.37x36 L272
7x38 7.39x38 I274
7x41 7.42x41 S277
7x42 7.43x42 H278
7x43 7.44x43 T279
7x45 7.45x45 N280
7x46 7.46x46 S281
7x47 7.47x47 V282
7x49 7.49x49 N284
H8
8x66 8.66x66 Q311
8x68 8.68x68 P313